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Synthesis of (+)-(1S)-1-pyrophosphoryl-(2R, 3R)-2,3-dihydroxy-(4S)-4-(phosphoryloxymethyl)cyclopentane, a stable, optically-active carbocyclic analog of 5-phosphoribosyl-1-pyrophosphate (PRPP) • ARTICLE Ronald J. Parry, Mark R. Burns, Sao Jiralerspong and Lawrence Alemany Abstract | Abstract + References | PDF (691 K) | |||
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Reaction of a 1-azirine-3-methylacrylate and derivatives with diphenylketene. A convenient route to 5-pyrrolin-2-ones • ARTICLE Albert Kascheres, José Nunes, Jr. and Fernando Brandão Abstract | Abstract + References | PDF (380 K) | |||
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The Knoevenagel condensation of O,S- and S,S-diethyl malonates and ethyl pyruvate • ARTICLE Bogdan K. Wilk Abstract | Abstract + References | PDF (229 K) | |||
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Fluorine-substituted derivatives of the carcinogenic dihydrodiol and diol epoxide metabolites of 7-methyl-, 12-methyl- and 7,12-dimethylbenz[a]anthracene • ARTICLE Ronald G. Harvey and Cecilia Cortez Abstract | Abstract + References | PDF (1112 K) | |||
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A simple, stereoselective synthesis of ketomethylene dipeptide isosteres • ARTICLE Robert V. Hoffman and Junhua Tao Abstract | Abstract + References | PDF (491 K) | |||
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Asymmetric synthesis of a taxol C-ring by aldol condensation and radical cyclization • ARTICLE David Crich, Xian-Yun Jiao and Milan Bruncko Abstract | Abstract + References | PDF (761 K) | |||
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Synthesis of the taxol AB-system by olefination of an A-ring C1 ketone and direct B-ring closure • ARTICLE David Crich, Swaminathan Natarajan and Joyce Z. Crich Abstract | Abstract + References | PDF (1395 K) | |||
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Fluorescent molecular probes I. The synthesis and biological properties of an ELF®  -glucuronidase substrate that yields fluorescent precipitates at the enzymatic activity sites • ARTICLEZhenjun Diwu, Yixin Lu, Rosalyn H. Upson, Mingjie Zhou, Dieter H. Klaubert and Richard P. Haugland Abstract | Abstract + References | PDF (371 K) | |||
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Photochemical reactions of sulfide-containing alkyl phenylglyoxylates • ARTICLE Shengkui Hu and Douglas C. Neckers Abstract | Abstract + References | PDF (860 K) | |||
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Purification of 9N-[(1′R,3′R)-trans-3′-hydroxycyclopentanyl]adenine HCl: a combination of theory and experiment • ARTICLE Robert Barbuch, Timothy T. Curran, David A Hay and Roy J. Vaz Abstract | Abstract + References | PDF (528 K) | |||
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Stereoselective reactions. 26. Solution structures of chiral bidentate lithium amide in relation to the solvent-dependent enantioselectivities in deprotonation reaction • ARTICLE Daisaku Sato, Hisashi Kawasaki, Ichio Shimada, Yoji Arata, Kimio Okamura, Tadamasa Date and Kenji Koga Abstract | Abstract + References | PDF (515 K) | |||
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Highly enantioselective cyclopropanation of styrene derivatives using Co(III)-salen complex as a catalyst • ARTICLE Tsutomu Fukuda and Tsutomu Katsuki Abstract | Abstract + References | PDF (474 K) | |||
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Total synthesis of (−)-periplanones C and D. Their pheromonal activities against three Periplaneta species • ARTICLE Yoshinori Nishii, Keisuke Watanabe, Taichi Yoshida, Tatsutoshi Okayama, Shozo Takahashi and Yoo Tanabe Abstract | Abstract + References | PDF (468 K) | |||
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Enantioselective synthesis of new C2-symmetric ferrocenylalkylamines via sonochemical amination of 1-ferrocenylalkyl acetates • ARTICLE Marcell Woltersdorf, Remo Kranich and Hans-Günther Schmalz Abstract | Abstract + References | PDF (687 K) | |||
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Protein mimetics (TASP) by sequential condensation of peptide loops to an immobilised topological template • ARTICLE Stéphane Peluso, Pascal Dumy, Ian M. Eggleston, Patrick Garrouste and Manfred Mutter Abstract | Abstract + References | PDF (364 K) | |||
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Preparation and reactions of new zincated nitrogen-containing heterocycles • ARTICLE A. S. Bhanu Prasad, Thomas M. Stevenson, Janakiram Rao Citineni, Valérie Nyzam and Paul Knochel Abstract | Abstract + References | PDF (1188 K) | |||
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Diastereoselective and convergent synthesis of both 11′-epimers of (−)-(2R,3R,6S)-carnavaline • ARTICLE Axel Pahl, Jörg Oetting, Jens Holzkamp and Hartmut H. Meyer Abstract | Abstract + References | PDF (742 K) | |||
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Synthesis of optically pure  -hydroxyglycine peptides • ARTICLEMichael Bogenstätter and Wolfgang Steglich Abstract | Abstract + References | PDF (426 K) | |||
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Synthesis of metallo--lactamase inhibitors • ARTICLE Magnus W. Walter, Robert M. Adlington, Jack E. Baldwin and Christopher J. Schofield Abstract | Abstract + References | PDF (987 K) | |||
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A new, effective approach for the C---C bond formation utilizing 1-,2- and 3-phosphonyl substituted radicals derived from iodoalkylphosphonates and n-Bu3SnH/Et3B/O2 system • ARTICLE Piotr Balczewski and Witold M. Pietrzykowski Abstract | Abstract + References | PDF (669 K) | |||
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Structure and absolute stereochemistry of the new cyclolinteinol and cyclolinteinol acetate, macrophage activation modulators • ARTICLE Alfonso Carotenuto, Ernesto Fattorusso, Virginia Lanzotti, Silvana Magno, Rosa Carnuccio and Fulvio D'Acquisto Abstract | Abstract + References | PDF (347 K) | |||
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Pyrrolidinamine, piperidinamine and tetrahydropyridazine derivatives from selenium promoted cyclization of alkenyl phenylhydrazones • ARTICLE Marcello Tiecco, Lorenzo Testaferri, Francesca Marini, Claudio Santi, Luana Bagnoli and Andrea Temperini Abstract | Abstract + References | PDF (380 K) | |||
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Chemical modifications on the acyclic moiety of 3-(2-hydroxyethoxy)-1-alkoxypropyl nucleobases. 2. Differentiation and growth inhibition in rhabdomyosarcoma cells after exposure to a novel 5-fluorouracil acyclonucleoside • ARTICLE Jose A. Gómez, Joaquín Campos, Juan A. Marchal, María A. Trujillo, Consolación Melguizo, José Prados, Miguel A. Gallo, Antonia Aránega and Antonio Espinosa Abstract | Abstract + References | PDF (1023 K) | |||
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Selective esterification of aliphatic nonconjugated carboxylic acids in the presence of aromatic or conjugated carboxylic acids catalysed by NiCl2.6H2O • ARTICLE Ram N. Ram and I. Charles Abstract | Abstract + References | PDF (285 K) | |||
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C---C bond fission via sulphones: A new ring cleavage of cyclic -keto phenylsulphones • ARTICLE Roberto Ballini, Giovanna Bosica and Tiziana Mecozzi Abstract | Abstract + References | PDF (230 K) | |||
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A chemical method for the preparation of novel 1,5-benzodiazepines acting as CCK-B antagonists in high enantiomeric purity • ARTICLE Giovanni Curotto, Daniele Donati, Gabriella Finizia and Antonella Ursini Abstract | Abstract + References | PDF (862 K) | |||
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Unusual reversal of stereoselectivity of 1,3-dipolar cycloaddition in the presence of Lewis acids • ARTICLE Philip C. Bulman Page, Mark Purdle and David Lathbury Abstract | Abstract + References | PDF (373 K) | |||
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Contributors to this issue • MISCELLANEOUS PDF (49 K) | |||
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Graphical abstracts • ABSTRACT PDF (341 K) | |||
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